CAS 1217459-13-6|3,3'-Diiodo-L-thyronine-13C6

Introduction:Basic information about CAS 1217459-13-6|3,3'-Diiodo-L-thyronine-13C6, including its chemical name, molecular formula, synonyms, physicochemical properties, and safety information, etc.
Common Name3,3'-Diiodo-L-thyronine-13C6
CAS Number1217459-13-6Molecular Weight531.03300
Density/Boiling Point/
Molecular FormulaC15H13I2NO4Melting Point/
MSDSChineseUSAFlash Point/
Symbol
GHS07
Signal WordWarning

Names

Name(2S)-2-amino-3-[4-(4-hydroxy-3-iodophenoxy)-3-iodophenyl]propanoic acid
SynonymMore Synonyms

3,3'-Diiodo-L-thyronine-13C6 BiologicalActivity

Description3,3'-Diiodo-L-thyronine-13C6 is the 13C labeled 3,3'-Diiodo-L-thyronine[1]. 3,3'-Diiodo-L-thyronine (3,3'-T2) is an endogenous metabolite of thyroid hormone. 3,3'-Diiodo-L-thyronine significantly enhances COX activity[2][3].
Related CatalogSignaling Pathways >>Immunology/Inflammation >>COXResearch Areas >>Metabolic Disease
In VitroStable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs[1].
References

[1]. Russak EM, et al. Impact of Deuterium Substitution on the Pharmacokinetics of Pharmaceuticals. Ann Pharmacother. 2019 Feb;53(2):211-216.  

[2]. Lorenzini L, et al. Assay of Endogenous 3,5-diiodo-L-thyronine (3,5-T2) and 3,3'-diiodo-L-thyronine (3,3'-T2) in Human Serum: A Feasibility Study. Front Endocrinol (Lausanne). 2019 Feb 19;10:88.  

[3]. Lanni A, et al. Rapid stimulation in vitro of rat liver cytochrome oxidase activity by 3,5-diiodo-L-thyronine and by 3,3'-diiodo-L-thyronine. Mol Cell Endocrinol. 1994 Feb99(1):89-94.  

[4]. Chen X, et al. Simultaneous quantification of T4, T3, rT3, 3,5-T2 and 3,3'-T2 in larval zebrafish (Danio rerio) as a model to study exposure to polychlorinated biphenyls. Biomed Chromatogr. 2018 Jun32(6):e4185.  

Chemical & Physical Properties

Molecular FormulaC15H13I2NO4
Molecular Weight531.03300
Exact Mass530.91400
PSA92.78000
LogP4.04840
InChIKeyCPCJBZABTUOGNM-USQDWSSZSA-N
SMILESNC(Cc1ccc(Oc2ccc(O)c(I)c2)c(I)c1)C(=O)O

Safety Information

Symbol
GHS07
Signal WordWarning
Hazard StatementsH302
RIDADRNONH for all modes of transport

Synonyms

3,3 inverted exclamation marka-Diiodo-L-thyronine-(phenoxy-13C6) (T2)
T2-13C6
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