CAS 516-72-3|20(S)-Hydroxycholesterol

Introduction:Basic information about CAS 516-72-3|20(S)-Hydroxycholesterol, including its chemical name, molecular formula, synonyms, physicochemical properties, and safety information, etc.
Common Name20(S)-Hydroxycholesterol
CAS Number516-72-3Molecular Weight402.65
Density1.03g/cm3Boiling Point512.3ºC at 760mmHg
Molecular FormulaC27H46O2Melting Point136-137ºC
MSDSChineseUSAFlash Point213.1ºC

Names

Name20-hydroxycholesterol
SynonymMore Synonyms

20(S)-Hydroxycholesterol BiologicalActivity

Description20(S)-hydroxyCholesterol (20α-Hydroxycholesterol) is an allosteric activator of the oncoprotein smoothened (Smo) that activates the hedgehog (Hh) signaling pathway with an EC50 of 3 μM in a gene transcription reporter assay using NIH3T3 cells[1][2].
Related CatalogSignaling Pathways >>Stem Cell/Wnt >>SmoResearch Areas >>Cancer
Target

EC50: 3 μM (hedgehog signaling pathway)[1]

References

[1]. Nachtergaele S, et al. Oxysterols are allosteric activators of the oncoprotein Smoothened. Nat Chem Biol. 2012 Jan 8;8(2):211-20.

[2]. Nedelcu D, et al, Oxysterol binding to the extracellular domain of Smoothened in Hedgehog signaling. Nat Chem Biol. 2013 Sep;9(9):557-64.

Chemical & Physical Properties

Density1.03g/cm3
Boiling Point512.3ºC at 760mmHg
Melting Point136-137ºC
Molecular FormulaC27H46O2
Molecular Weight402.65
Flash Point213.1ºC
Exact Mass402.35000
PSA40.46000
LogP6.50360
Index of Refraction1.538
InChIKeyMCKLJFJEQRYRQT-APGJSSKUSA-N
SMILESCC(C)CCCC(C)(O)C1CCC2C3CC=C4CC(O)CCC4(C)C3CCC21C
Storage condition-20°C Freezer

Safety Information

Personal Protective EquipmentEyeshields;Gloves;type N95 (US);type P1 (EN143) respirator filter
Hazard CodesXi
RIDADRNONH for all modes of transport
WGK Germany3

Articles29

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Human adipose-derived stem cells have been identified as a potential source of cells for use in bone tissue engineering because of their ready availability, ease of harvest, and susceptibility to oste...

Conversion of exogenous cholesterol into glycoalkaloids in potato shoots, using two methods for sterol solubilisation.

PLoS ONE 8 , e82955, (2013)

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Oxpholipin 11D: an anti-inflammatory peptide that binds cholesterol and oxidized phospholipids.

PLoS ONE 5 , e10181, (2010)

Many gram-positive bacteria produce pore-forming exotoxins that contain a highly conserved, 12-residue domain (ECTGLAWEWWRT) that binds cholesterol. This domain is usually flanked N-terminally by argi...

Synonyms

20α-Hydroxy Cholesterol
20ALPHA-HYDROXYCHOLESTEROL
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