Introduction：Basic information about CAS 202591-23-9|CPI-203, including its chemical name, molecular formula, synonyms, physicochemical properties, and safety information, etc.
| Common Name | CPI-203 |
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| CAS Number | 202591-23-9 | Molecular Weight | 399.897 |
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| Density | 1.5±0.1 g/cm3 | Boiling Point | 690.5±65.0 °C at 760 mmHg |
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| Molecular Formula | C19H18ClN5OS | Melting Point | / |
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| MSDS | / | Flash Point | 371.4±34.3 °C |
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Names
| Name | 2-[(6S)-4-(4-Chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl]acetamide |
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| Synonym | More Synonyms |
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CPI-203 BiologicalActivity
| Description | (Rac)-CPI-203 is a racemate of CPI-203 (HY-15846) (BET bromodomain inhibitor)[1] |
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| Related Catalog | Research Areas >>CancerSignaling Pathways >>Others >>Others |
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| References | [1]. Moros A, et al. Synergistic antitumor activity of lenalidomide with the BET bromodomain inhibitor CPI203 in bortezomib-resistant mantle cell lymphoma. Leukemia. 2014 Oct;28(10):2049-59 |
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Chemical & Physical Properties
| Density | 1.5±0.1 g/cm3 |
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| Boiling Point | 690.5±65.0 °C at 760 mmHg |
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| Molecular Formula | C19H18ClN5OS |
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| Molecular Weight | 399.897 |
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| Flash Point | 371.4±34.3 °C |
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| Exact Mass | 399.092072 |
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| LogP | 1.85 |
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| Vapour Pressure | 0.0±2.2 mmHg at 25°C |
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| Index of Refraction | 1.749 |
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| InChIKey | QECMENZMDBOLDR-UHFFFAOYSA-N |
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| SMILES | Cc1sc2c(c1C)C(c1ccc(Cl)cc1)=NC(CC(N)=O)c1nnc(C)n1-2 |
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| Storage condition | 2-8℃ |
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Synonyms
| 2-[(6S)-4-(4-Chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl]acetamide |
| 6H-Thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetamide, 4-(4-chlorophenyl)-2,3,9-trimethyl-, (6S)- |
| 4-(4-Chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetamide |
| CPI-203 |
