CAS 10140-70-2|Curvularin

Introduction:Basic information about CAS 10140-70-2|Curvularin, including its chemical name, molecular formula, synonyms, physicochemical properties, and safety information, etc.
Common NameCurvularin
CAS Number10140-70-2Molecular Weight292.32700
Density1.2g/cm3Boiling Point557ºC at 760mmHg
Molecular FormulaC16H20O5Melting Point205-207 °C
MSDSChineseUSAFlash Point207.9ºC
Symbol
GHS07
Signal WordWarning

Names

Name2H-3-Benzoxacyclododecin-2,10(1H)-dione, 4,5,6,7,8,9-hexahydro-11,13-dihydroxy-4-methyl-, (-)
SynonymMore Synonyms

Curvularin BiologicalActivity

DescriptionCurvularin, a fungal metabolite and a potent mycotoxin naturally isolated from Curvularia lunata, inhibits cytokine-induced nitric oxide synthase (iNOS), with an IC50 of 9.5 µM[1][2].
Related CatalogResearch Areas >>OthersSignaling Pathways >>Immunology/Inflammation >>NO Synthase
Target

IC50: 9.5 µM (iNOS)[2].

References

[1]. Kumar CG, et al. Metabolite profiling and biological activities of bioactive compounds produced by Chrysosporium lobatum strain BK-3 isolated from Kaziranga National Park, Assam, India. Springerplus. 2013 Dec;2(1):122.

[2]. Yao Y, et al. Sporogen, S14-95, and S-curvularin, three inhibitors of human inducible nitric-oxide synthase expression isolated from fungi. Mol Pharmacol. 2003 Feb;63(2):383-91.

Chemical & Physical Properties

Density1.2g/cm3
Boiling Point557ºC at 760mmHg
Melting Point205-207 °C
Molecular FormulaC16H20O5
Molecular Weight292.32700
Flash Point207.9ºC
Exact Mass292.13100
PSA83.83000
LogP2.71880
Vapour Pressure5.18E-13mmHg at 25°C
Index of Refraction1.54
InChIKeyVDUIGYAPSXCJFC-JTQLQIEISA-N
SMILESCC1CCCCCC(=O)c2c(O)cc(O)cc2CC(=O)O1

Safety Information

Symbol
GHS07
Signal WordWarning
Hazard StatementsH302
Hazard CodesXn
RIDADRNONH for all modes of transport

Articles15

More Articles
Sulfur-containing cytotoxic curvularin macrolides from Penicillium sumatrense MA-92, a fungus obtained from the rhizosphere of the mangrove Lumnitzera racemosa.

J. Nat. Prod. 76(11) , 2145-9, (2013)

Sumalarins A-C (1-3), the new and rare examples of sulfur-containing curvularin derivatives, along with three known analogues (4-6), were isolated and identified from the cytotoxic extract of Penicill...

Metabolite production by differentUlocladiumspecies

Int. J. Food Microbiol. 126(1-2) , 172-9, (2008)

Ulocladium, which is phylogenetically related to Alternaria, contains species that are food spoilers and plant pathogens, but also species that have potential as enzyme producers and bio-control agent...

[Molecular basis of probes for cytoskeletal proteins].

Tanpakushitsu Kakusan Koso. 38(11) , 1730-41, (1993)

Synonyms

curvularin
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