CAS 75184-71-3|Albendazole sulfone

Introduction:Basic information about CAS 75184-71-3|Albendazole sulfone, including its chemical name, molecular formula, synonyms, physicochemical properties, and safety information, etc.
Common NameAlbendazole sulfone
CAS Number75184-71-3Molecular Weight297.33000
Density1.42g/cm3Boiling Point/
Molecular FormulaC12H15N3O4SMelting Point290-292ºC
MSDSChineseUSAFlash Point/
Symbol
GHS07, GHS08
Signal WordWarning

Names

NameAlbendazole sulfone
SynonymMore Synonyms

Albendazole sulfone BiologicalActivity

DescriptionAlbendazole sulfone is a metabolite of Albendazole, and exhibits anti-parasite effect against Echinococcus multilocularis Metacestodes[1][2].
Related CatalogResearch Areas >>Infection
References

[1]. Ingold K, et, al. Efficacies of albendazole sulfoxide and albendazole sulfone against In vitro-cultivated Echinococcus multilocularis metacestodes. Antimicrob Agents Chemother. 1999 May;43(5):1052-61.

[2]. Adas G, et, al. Use of albendazole sulfoxide, albendazole sulfone, and combined solutions as scolicidal agents on hydatid cysts (in vitro study). World J Gastroenterol. 2009 Jan 7;15(1):112-6.

Chemical & Physical Properties

Density1.42g/cm3
Melting Point290-292ºC
Molecular FormulaC12H15N3O4S
Molecular Weight297.33000
Exact Mass297.07800
PSA109.53000
LogP3.07870
Index of Refraction1.619
InChIKeyCLSJYOLYMZNKJB-UHFFFAOYSA-N
SMILESCCCS(=O)(=O)c1ccc2nc(NC(=O)OC)[nH]c2c1
Storage condition-20°C Freezer
Water SolubilitySoluble in DMSO, and methanol.

Toxicological Information

CHEMICAL IDENTIFICATION

RTECS NUMBER :
DD6520700
CHEMICAL NAME :
2-Benzimidazolecarbamic acid, 5-(propylsulfonyl)-, methyl ester
CAS REGISTRY NUMBER :
75184-71-3
LAST UPDATED :
198910
DATA ITEMS CITED :
2
MOLECULAR FORMULA :
C12-H15-N3-O4-S
MOLECULAR WEIGHT :
297.36
WISWESSER LINE NOTATION :
T56 BM DNJ CMVO1 GSW3

HEALTH HAZARD DATA

ACUTE TOXICITY DATA

TYPE OF TEST :
TDLo - Lowest published toxic dose
ROUTE OF EXPOSURE :
Oral
DOSE :
75 mg/kg
SEX/DURATION :
female 8-15 day(s) after conception
TOXIC EFFECTS :
Reproductive - Effects on Embryo or Fetus - fetotoxicity (except death, e.g., stunted fetus) Reproductive - Effects on Embryo or Fetus - fetal death Reproductive - Specific Developmental Abnormalities - musculoskeletal system
REFERENCE :
ARCVBP Annales Recherches Veterinaires. (Institut National de la Recherche Agronomique, Service des Publ., Route de Saint-Cyr, 78000 Versailles, France) V.1- 1970- Volume(issue)/page/year: 12,159,1981
TYPE OF TEST :
TDLo - Lowest published toxic dose
ROUTE OF EXPOSURE :
Oral
DOSE :
75 mg/kg
SEX/DURATION :
female 8-15 day(s) after conception
TOXIC EFFECTS :
Reproductive - Specific Developmental Abnormalities - other developmental abnormalities
REFERENCE :
ARCVBP Annales Recherches Veterinaires. (Institut National de la Recherche Agronomique, Service des Publ., Route de Saint-Cyr, 78000 Versailles, France) V.1- 1970- Volume(issue)/page/year: 12,159,1981

Safety Information

Symbol
GHS07, GHS08
Signal WordWarning
Hazard StatementsH315-H319-H361d
Precautionary StatementsP281-P305 + P351 + P338
Hazard CodesXn
Risk Phrases63-36/38
Safety Phrases26-36/37
RIDADRNONH for all modes of transport
RTECSDD6520700
HS Code29339900

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Synonyms

albendazole sulfone
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