CAS 6018-19-5|Sodium 4-aminosalicylate dihydrate

Introduction:Basic information about CAS 6018-19-5|Sodium 4-aminosalicylate dihydrate, including its chemical name, molecular formula, synonyms, physicochemical properties, and safety information, etc.
Common NameSodium 4-aminosalicylate dihydrate
CAS Number6018-19-5Molecular Weight211.148
Density/Boiling Point380.8ºC at 760 mmHg
Molecular FormulaC7H10NNaO5Melting Point250 °C
MSDSChineseUSAFlash Point184.1ºC
Symbol
GHS07
Signal WordWarning

Names

NameSodium 4-aminosalicylate dihydrate
SynonymMore Synonyms

Sodium 4-aminosalicylate dihydrate BiologicalActivity

DescriptionSodium 4-aminosalicylate dihydrate is one of the antimycobacterial drugs currently used for multidrug-resistant tuberculosis.
Related CatalogSignaling Pathways >>Anti-infection >>BacterialResearch Areas >>Infection
References

[1]. Zheng J, et al. para-Aminosalicylic acid is a prodrug targeting dihydrofolate reductase in Mycobacterium tuberculosis. J Biol Chem. 2013 Aug 9;288(32):23447-56.

[2]. Sy SK, et al. N-acetyltransferase genotypes and the pharmacokinetics and tolerability of para-aminosalicylic acid in drug-resistant pulmonary tuberculosis patients. Antimicrob Agents Chemother. 2015 May 11. pii: AAC.04049-14.

Chemical & Physical Properties

Boiling Point380.8ºC at 760 mmHg
Melting Point250 °C
Molecular FormulaC7H10NNaO5
Molecular Weight211.148
Flash Point184.1ºC
Exact Mass211.045670
PSA104.84000
InChIKeyGMUQJDAYXZXBOT-UHFFFAOYSA-M
SMILESNc1ccc(C(=O)[O-])c(O)c1.O.O.[Na+]
Water Solubilitysoluble

Safety Information

Symbol
GHS07
Signal WordWarning
Hazard StatementsH315-H319-H335
Precautionary StatementsP305 + P351 + P338
Personal Protective Equipmentdust mask type N95 (US);Eyeshields;Gloves
Hazard CodesXi: Irritant;
Risk PhrasesR36/37/38
Safety PhrasesS26-S36
RIDADRNONH for all modes of transport
WGK Germany3
HS Code2918219000

Customs

HS Code2922509090
Summary2922509090. other amino-alcohol-phenols, amino-acid-phenols and other amino-compounds with oxygen function. VAT:17.0%. Tax rebate rate:13.0%. . MFN tariff:6.5%. General tariff:30.0%

Articles26

More Articles
Adsorption of phenolic compounds from aqueous solution using salicylic acid type adsorbent.

J. Hazard. Mater. 201-202 , 74-81, (2012)

In this study, 5-aminosalicylic acid (5-ASA) was successfully grafted onto the poly(glycidyl methacrylate) (PGMA) macromolecular chains of PGMA/SiO(2) to obtain adsorbent ASA-PGMA/SiO(2). The adsorpti...

Comparison between 5-aminosalicylic acid (5-ASA) and para-aminosalicylic acid (4-PAS) as potential protectors against Mn-induced neurotoxicity.

Biol. Trace Elem. Res. 152(1) , 113-6, (2013)

Manganese (Mn) is an essential metal for biological systems; however, occupational or clinical exposure to high levels of Mn can produce a neurological disorder called manganism. Oxidative stress and ...

Liver-selective expression of human arylamine N-acetyltransferase NAT2 in transgenic mice.

Drug Metab. Dispos. 39(5) , 882-90, (2011)

Human arylamine N-acetyltransferase 2 (NAT2) mediates the biotransformation of arylamine drugs and procarcinogens into either innocuous or reactive DNA-damaging metabolites and is expressed predominan...

Synonyms

Sodium 4-Aminosalicylate
EINECS 205-091-2
4-amino-2-hydroxybenzoic acid sodium salt dihydrate
Benzoic acid, 4-amino-2-hydroxy-, monosodium salt, dihydrate
Benzoic acid, 4-amino-2-hydroxy-, sodium salt, hydrate (1:1:2)
4-Aminosalicylic acid sodium salt dihydrate
AMINOSALICYLATE SODIUM,DIHYDRATE
4-AMINOSALICYLIC ACID,NA SALT
Sodium 4-amino-2-hydroxybenzoate dihydrate
4-AMINOSALICYLIC ACID SODIUM SALT 2-HYDRATE
4-Amino-2-hydroxy-benzoesaeure,Natrium-Salz
4-AMINOSALICYLIC ACID SODIUM DIHYDRATE
sodium p-aminosalicylate dihydrate
SODIUM AMINOSALICYLA
4-amino-2-hydroxy-benzoic acid,sodium-salt
4-amino-salicylic acid sodium salt
AMINOSALICYLATESODIUM,DIHYDRATE,USP
UNII-S38B9W6AXW
PAS-NA 2H2O
Sodium 4-aminosalicy
MFCD00151044
Sodium 4-amino-2-hydroxybenzoate hydrate (1:1:2)
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