CAS 1001415-66-2|Remimazolam benzenesulfonate

Introduction：Basic information about CAS 1001415-66-2|Remimazolam benzenesulfonate, including its chemical name, molecular formula, synonyms, physicochemical properties, and safety information, etc.

Table of Contents

1. Names
2. Remimazolam benzenesulfonate BiologicalActivity
3. Chemical & Physical Properties
4. Synonyms

Common Name	Remimazolam benzenesulfonate
CAS Number	1001415-66-2	Molecular Weight	597.48000
Density	/	Boiling Point	/
Molecular Formula	C₂₇H₂₅BrN₄O₅S	Melting Point	/
MSDS	/	Flash Point	/

Names

Name	Remimazolam benzenesulfonate
Synonym	More Synonyms

Remimazolam benzenesulfonate BiologicalActivity

Description	Remimazolam benzenesulfonate is a GABA agonist。Target: GABA ReceptorRemimazolam acts on GABA receptor, specifically GABA-alpha. Remimazolam is a new drug innovation in anesthesia. Remimazolam combines the properties of two unique drugs already established in anesthesia - Midazolam and remifentanil. Remimazolam acts on GABA receptors like midazolam and has organ-independent metabolism like remifentanil. Remimazolam is likely to be the sedative of the future, as preliminary phase II trials have shown minimal residual effects on prolonged infusions. Remimazolam has potential to be used as a sedative in ICU and as a novel agent for procedural sedation.
Related Catalog	Signaling Pathways >>Membrane Transporter/Ion Channel >>GABA ReceptorSignaling Pathways >>Neuronal Signaling >>GABA ReceptorResearch Areas >>Neurological Disease
References	[1]. Goudra BG, et al. Remimazolam: The future of its sedative potential. Saudi J Anaesth. 2014 Jul;8(3):388-391.

Chemical & Physical Properties

Molecular Formula	C₂₇H₂₅BrN₄O₅S
Molecular Weight	597.48000
Exact Mass	596.07300
PSA	132.12000
LogP	5.63320
InChIKey	QMTKNJZIWGTNTE-LMOVPXPDSA-N
SMILES	COC(=O)CCC1N=C(c2ccccn2)c2cc(Br)ccc2-n2c(C)cnc21.O=S(=O)(O)c1ccccc1
Storage condition	2-8℃

Synonyms

CN-7056 benzenesulfonate

methyl (S)-3-(8-bromo-1-methyl-6-(pyridin-2-yl)-4H-benzo[f]imidazo[1,2-a][1,4]diazepin-4-yl)propanoate benzenesulfonate

Remimazolam (benzenesulfonate)

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