CAS 17355-11-2|Tyr-Phe

Introduction:Basic information about CAS 17355-11-2|Tyr-Phe, including its chemical name, molecular formula, synonyms, physicochemical properties, and safety information, etc.
Common NameTyr-Phe
CAS Number17355-11-2Molecular Weight328.36200
Density1.3 g/cm3Boiling Point642.2ºC at 760 mmHg
Molecular FormulaC18H20N2O4Melting Point/
MSDSChineseUSAFlash Point342.2ºC

Names

Name2-[[2-amino-3-(4-hydroxyphenyl)propanoyl]amino]-3-phenylpropanoic acid
SynonymMore Synonyms

Tyr-Phe BiologicalActivity

DescriptionH-Tyr-Phe-OH (L-Tyrosyl-L-phenylalanine) is an orally active inhibitor of Angiotensin converting enzyme (ACE), with an inhibiton rate of 48% at 50 μM. H-Tyr-Phe-OH can be used as an biomarker for differentiating benign thyroid nodules (BTN) from thyroid cancer (TC). H-Tyr-Phe-OH exhibits xanthine oxidase inhibition (uric acid lowering) activity and serves as regulator in IL-8 production in neutrophil-like cells[1][2][3][4].
Related CatalogResearch Areas >>CancerSignaling Pathways >>Metabolic Enzyme/Protease >>Angiotensin-converting Enzyme (ACE)Research Areas >>Inflammation/ImmunologySignaling Pathways >>Metabolic Enzyme/Protease >>Xanthine Oxidase
Target

Target: ACE (Angiotensin converting enzyme), xanthine oxidase[1]

References

[1]. Zhu Wei, et al. Biomarker containing keratin type II cytoskeleton 1b for differentiating benign thyroid nodules and thyroid cancer: China, CN114264828A[P]. 2022-04-01.

[2]. Enari Hiroyuki, et al. Angiotensin converting enzyme (ACE)-inhibiting peptides, ACE inhibitors containing the peptides, their uses, and manufacture of the peptides from shark cartilage: Japan, JP2005154326A[P]. 2005-06-16.

[3]. Mao Xiangchao, et al. Method for preparing cod fish peptide with xanthine oxidase inhibitory activity: China, CN113005166A[P]. 2021-06-22.

[4]. Hsueh PC, et al. Metabolomic profiling of parapneumonic effusion reveals a regulatory role of dipeptides in interleukin-8 production in neutrophil-like cells. Anal Chim Acta. 2020 Sep 1;1128:238-250.

Chemical & Physical Properties

Density1.3 g/cm3
Boiling Point642.2ºC at 760 mmHg
Molecular FormulaC18H20N2O4
Molecular Weight328.36200
Flash Point342.2ºC
Exact Mass328.14200
PSA112.65000
LogP2.16530
Vapour Pressure2.27E-17mmHg at 25°C
Index of Refraction1.625
InChIKeyCGWAPUBOXJWXMS-HOTGVXAUSA-N
SMILESNC(Cc1ccc(O)cc1)C(=O)NC(Cc1ccccc1)C(=O)O

Safety Information

Personal Protective EquipmentEyeshields;Gloves;type N95 (US);type P1 (EN143) respirator filter
RIDADRNONH for all modes of transport
HS Code2924299090

Customs

HS Code2924299090
Summary2924299090. other cyclic amides (including cyclic carbamates) and their derivatives; salts thereof. VAT:17.0%. Tax rebate rate:13.0%. . MFN tariff:6.5%. General tariff:30.0%

Articles3

More Articles
A new cytochrome C reducing dipeptide.

J. Natl. Med. Assoc. 82 , 113-116, (1990)

Using absorption spectroscopy, it has been found that tyrosylphenylalanine specifically reduces cytochrome C. This effect is pH and concentration dependent with the EC +/- SE = 4.42 x 10(-3) M. At 10(...

The effect of neighboring methionine residue on tyrosine nitration and oxidation in peptides treated with MPO, H2O2, and NO2(-) or peroxynitrite and bicarbonate: role of intramolecular electron transfer mechanism?

Arch. Biochem. Biophys. 484 , 134-145, (2009)

Recent reports suggest that intramolecular electron transfer reactions can profoundly affect the site and specificity of tyrosyl nitration and oxidation in peptides and proteins. Here we investigated ...

Interaction between cytochrome C and di- and tripeptides.

Life Sci. 48 , 523-530, (1991)

By observing changes in the absorbance spectrum between 340 and 650 nm, we found that tyrosyltyrosylphenylalanine (TTP) interacts with cytochrome C (CC). TTP caused the characteristic changes of CC re...

Synonyms

H-Tyr-Phe-OH
Tyr-Phe
L-tyrosyl-L-phenylalanine
tyrosylphenylalanine
tyrosinylphenylalanine
L-Tyrosine-L-phenylalanine
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