CAS 3443-84-3|2-Oleoylglycerol

Introduction:Basic information about CAS 3443-84-3|2-Oleoylglycerol, including its chemical name, molecular formula, synonyms, physicochemical properties, and safety information, etc.
Common Name2-Oleoylglycerol
CAS Number3443-84-3Molecular Weight356.54000
Density0.969 g/cm3Boiling Point485.4ºC at 760mmHg
Molecular FormulaC21H40O4Melting Point/
MSDSChineseUSAFlash Point113ºC

Names

Name2-oleoylglycerol
SynonymMore Synonyms

2-Oleoylglycerol BiologicalActivity

Description2-Oleoylglycerol is a dietary naturally occurring lipid. 2-Oleoylglycerol is a GPR119 agonist, with an EC50 of 2.5 μM for human GPR119 in transiently transfected COS-7 cells. 2-Oleoylglycerol stimulates glucagon-like peptide-1 (GLP-1) secretion in vivo[1][2].
Related CatalogSignaling Pathways >>GPCR/G Protein >>GPR119Research Areas >>Metabolic Disease
Target

IC50: 2.5 μM (hGPR119) (in COS-7 cells)[1]

References

[1]. Hansen KB, et, al. 2-Oleoyl glycerol is a GPR119 agonist and signals GLP-1 release in humans. J Clin Endocrinol Metab. 2011 Sep;96(9):E1409-17.

[2]. Ghafouri N, et, al. Inhibition of monoacylglycerol lipase and fatty acid amide hydrolase by analogues of 2-arachidonoylglycerol. Br J Pharmacol. 2004 Nov;143(6):774-84.

Chemical & Physical Properties

Density0.969 g/cm3
Boiling Point485.4ºC at 760mmHg
Molecular FormulaC21H40O4
Molecular Weight356.54000
Flash Point113ºC
Exact Mass356.29300
PSA66.76000
LogP4.92030
Index of Refraction1.478
InChIKeyUPWGQKDVAURUGE-KTKRTIGZSA-N
SMILESCCCCCCCCC=CCCCCCCCC(=O)OC(CO)CO

Safety Information

Personal Protective EquipmentEyeshields;Gloves;type N95 (US);type P1 (EN143) respirator filter
RIDADRNONH for all modes of transport
WGK Germany3

Articles15

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Synonyms

glycerine monooleate
2-o-Kresyloxy-glutarsaeure-diethylester
2-MONOOLEIN
1,3-dihydroxypropan-2-yl oleate
2-monooleoylglycerol
2-Oleoylglycerol
glycerin oleate
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