CAS 64294-95-7|Setastine

Introduction：Basic information about CAS 64294-95-7|Setastine, including its chemical name, molecular formula, synonyms, physicochemical properties, and safety information, etc.

Table of Contents

1. Names
2. Setastine BiologicalActivity
3. Chemical & Physical Properties
4. Safety Information
5. Customs
6. Synonyms

Common Name	Setastine
CAS Number	64294-95-7	Molecular Weight	357.91700
Density	/	Boiling Point	/
Molecular Formula	C₂₂H₂₈ClNO	Melting Point	/
MSDS	/	Flash Point	/

Names

Name	1-[2-[1-(4-chlorophenyl)-1-phenylethoxy]ethyl]azepane
Synonym	More Synonyms

Setastine BiologicalActivity

Description	Setastine (EGIS-2062 (free acid); EGYT-2062 (free acid) is an orally effective, non-sedative and long acting anti-allergic agent. Setastine possesses potent histamine Hi-receptor blocking properties and can be used for allergies and rhinitis research[1]<.
Related Catalog	Signaling Pathways >>Immunology/Inflammation >>Histamine ReceptorResearch Areas >>Inflammation/ImmunologySignaling Pathways >>GPCR/G Protein >>Histamine Receptor
Target	IC50:Histamine Hi-receptor[1]
References	[1]. Németh, A., & Huszti, Z. (1988). The effect of a new antihistamine drug, Loderix® (EGIS-2062), on stimulus-evoked histamine release from rat peritoneal mast cells. Agents and Actions, 23(3-4), 194–197.

Chemical & Physical Properties

Molecular Formula	C₂₂H₂₈ClNO
Molecular Weight	357.91700
Exact Mass	357.18600
PSA	12.47000
LogP	5.43400
InChIKey	VBSPHZOBAOWFCL-UHFFFAOYSA-N
SMILES	CC(OCCN1CCCCCC1)(c1ccccc1)c1ccc(Cl)cc1

Safety Information

HS Code	2933990090

Customs

HS Code	2933990090
Summary	2933990090. heterocyclic compounds with nitrogen hetero-atom(s) only. VAT:17.0%. Tax rebate rate:13.0%. . MFN tariff:6.5%. General tariff:20.0%

Synonyms

1H-Azepine,1-(2-(1-(4-chlorophenyl)-1-phenylethoxy)ethyl)hexahydro

Setastine

Setastine [INN]

Setastina

Setastinum

1-(2-(1-(4-Chlorophenyl)-1-phenylethoxy)ethyl)azepane

Setastinum [INN-Latin]

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