CAS 452-06-2|2-Aminopurine

Introduction:Basic information about CAS 452-06-2|2-Aminopurine, including its chemical name, molecular formula, synonyms, physicochemical properties, and safety information, etc.
Common Name2-Aminopurine
CAS Number452-06-2Molecular Weight135.127
Density1.9±0.1 g/cm3Boiling Point328.2±25.0 °C at 760 mmHg
Molecular FormulaC5H5N5Melting Point280-282 °C(lit.)
MSDSChineseUSAFlash Point152.3±23.2 °C
Symbol
GHS07
Signal WordWarning

Names

Name2-aminopurine
SynonymMore Synonyms

2-Aminopurine BiologicalActivity

Description2-Aminopurine, a fluorescent analog of guanosine and adenosine, is a widely used fluorescence-decay-based probe of DNA structure. When 2-Aminopurine is inserted in anoligonucleotide, its fluorescence is highly quenched by stacking with the natural bases. 2-Aminopurine has been used to probe nucleic acid structure and dynamics[1][2].
Related CatalogResearch Areas >>OthersSignaling Pathways >>Others >>Others
In Vitro2-Aminopurine (2AP) is not valuable as afluorescent label because its fluorescence is highly quenched by stacking with the natural bases, when it is inserted in anoligonucleotide. However, it is this very susceptibility to interbase quenching that makes 2AP an exquisitely sensitivefluorescent probe of nucleic acid structure[1]. 2-Aminopurine differs from adenine (6-aminopurine) only in the position of the exocyclic amine group, and yet its fluorescence intensity is one thousand times that of adenine[1].
References

[1]. J M Jean, et al. 2-Aminopurine fluorescence quenching and lifetimes: role of base stacking. Proc Natl Acad Sci U S A. 2001 Jan 2;98(1):37-41.

[2]. Dehong Tan, et al. Decreased glycation and structural protection properties of γ-glutamyl-S-allyl-cysteine peptide isolated from fresh garlic scales (Allium sativum L.). Nat Prod Res. 2015;29(23):2219-22.

Chemical & Physical Properties

Density1.9±0.1 g/cm3
Boiling Point328.2±25.0 °C at 760 mmHg
Melting Point280-282 °C(lit.)
Molecular FormulaC5H5N5
Molecular Weight135.127
Flash Point152.3±23.2 °C
Exact Mass135.054489
PSA80.48000
LogP-1.33
Vapour Pressure0.0±0.7 mmHg at 25°C
Index of Refraction1.954
InChIKeyMWBWWFOAEOYUST-UHFFFAOYSA-N
SMILESNc1ncc2[nH]cnc2n1

Toxicological Information

CHEMICAL IDENTIFICATION

RTECS NUMBER :
UO7475000
CHEMICAL NAME :
Purine, 2-amino-
CAS REGISTRY NUMBER :
452-06-2
LAST UPDATED :
199612
DATA ITEMS CITED :
28
MOLECULAR FORMULA :
C5-H5-N5
MOLECULAR WEIGHT :
135.15
WISWESSER LINE NOTATION :
T56 BN DM FN HNJ GZ

HEALTH HAZARD DATA

ACUTE TOXICITY DATA

TYPE OF TEST :
LD50 - Lethal dose, 50 percent kill
ROUTE OF EXPOSURE :
Oral
SPECIES OBSERVED :
Rodent - rat
DOSE/DURATION :
723 mg/kg
TOXIC EFFECTS :
Details of toxic effects not reported other than lethal dose value
TYPE OF TEST :
LD50 - Lethal dose, 50 percent kill
ROUTE OF EXPOSURE :
Intraperitoneal
SPECIES OBSERVED :
Rodent - rat
DOSE/DURATION :
270 mg/kg
TOXIC EFFECTS :
Details of toxic effects not reported other than lethal dose value
TYPE OF TEST :
Specific locus test

MUTATION DATA

TYPE OF TEST :
Mutation in mammalian somatic cells
TEST SYSTEM :
Rodent - hamster Embryo
DOSE/DURATION :
100 mg/L
REFERENCE :
PNASA6 Proceedings of the National Academy of Sciences of the United States of America. (National Academy of Sciences, Printing & Pub. Office, 2101 Constitution Ave., Washington, DC 20418) V.1- 1915- Volume(issue)/page/year: 78,5685,1981

Safety Information

Symbol
GHS07
Signal WordWarning
Hazard StatementsH302
Precautionary StatementsP301 + P312 + P330
Personal Protective Equipmentdust mask type N95 (US);Eyeshields;Gloves
Hazard CodesXn:Harmful;
Risk PhrasesR22
Safety PhrasesS22-S36
RIDADRNONH for all modes of transport
WGK Germany3
RTECSUO7475000
HS Code2933990090

Customs

HS Code2933990090
Summary2933990090. heterocyclic compounds with nitrogen hetero-atom(s) only. VAT:17.0%. Tax rebate rate:13.0%. . MFN tariff:6.5%. General tariff:20.0%

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Synonyms

2-Aminoperin
iso-Adenine
2-Aminopurine
3H-Purin-2-amine
MFCD07357244
7H-Purin-2-amine
9H-Purin-2-amine
2-amino purine
EINECS 207-197-4
9H-purin-2-ylamine
Purine, 2-amino-
2-amino-6-purine
1H-Purin-2-amine
4-aminopurine
2-amino-purin
SQ 22,451
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