CAS 134678-17-4|Lamivudine

Introduction:Basic information about CAS 134678-17-4|Lamivudine, including its chemical name, molecular formula, synonyms, physicochemical properties, and safety information, etc.
Common NameLamivudine
CAS Number134678-17-4Molecular Weight229.256
Density1.7±0.1 g/cm3Boiling Point475.4±55.0 °C at 760 mmHg
Molecular FormulaC8H11N3O3SMelting Point177 °C
MSDSChineseUSAFlash Point241.3±31.5 °C
Symbol
GHS08
Signal WordWarning

Names

Namelamivudine
SynonymMore Synonyms

Lamivudine BiologicalActivity

DescriptionLamivudine is a nucleoside reverse transcriptase inhibitors?(NRTIs). Lamivudine can inhibit HIV reverse transcriptase 1/2 and also the reverse transcriptase of hepatitis B virus.
Related CatalogSignaling Pathways >>Anti-infection >>HIVSignaling Pathways >>Anti-infection >>Reverse TranscriptaseResearch Areas >>Infection
References

[1]. Li, Y.C., [A clinical study on lamivudine treatment for advanced schistosomisis with chronic B hepatits]. Zhongguo Xue Xi Chong Bing Fang Zhi Za Zhi, 2013. 25(5): p. 548-9, 551.

[2]. Zhang, C.E., et al., [Effects of lamivudine on growth of intestinal characteristic bacteria by microcalorimetry in vitro]. Yao Xue Xue Bao, 2013. 48(10): p. 1590-4.

Chemical & Physical Properties

Density1.7±0.1 g/cm3
Boiling Point475.4±55.0 °C at 760 mmHg
Melting Point177 °C
Molecular FormulaC8H11N3O3S
Molecular Weight229.256
Flash Point241.3±31.5 °C
Exact Mass229.052109
PSA115.67000
LogP-0.71
Vapour Pressure0.0±2.7 mmHg at 25°C
Index of Refraction1.755
InChIKeyJTEGQNOMFQHVDC-NKWVEPMBSA-N
SMILESNc1ccn(C2CSC(CO)O2)c(=O)n1
Storage conditionFreezer

Safety Information

Symbol
GHS08
Signal WordWarning
Hazard StatementsH361
Precautionary StatementsP281
Hazard CodesXi
Risk Phrases63
RIDADRNONH for all modes of transport
RTECSUW7361333
HS Code2934999090

Customs

HS Code2938901000
SummaryHS: 2938901000. 4-amino-1-((2r,5s)-2-(hydroxymethyl)-1,3-oxathiolan-5-yl)pyrimidin-2(1h)-one. VAT:17.0%. tax rebate rate:13.0%. supervision conditions:None. MFN tarrif:6.5%. general tariff:20.0%

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Synonyms

2(1H)-Pyrimidinone, 4-amino-1-[(2R,5S)-2-(hydroxymethyl)-1,3-oxathiolan-5-yl]-
3TC
Heptodin
cent
(-)-1-[(2R,5S)-2-(Hydroxymethyl)-1,3-oxathiolan-5-yl]cytosine
Lamivudine
Zeffix
Zefix
Hepitec
Heptivir
2(1H)-Pyrimidinone, 4-amino-1-[2-(hydroxymethyl)-1,3-oxathiolan-5-yl], (-)(2R,5S)
2',3'-Dideoxy-3'-thiacytidine
Heptovir
4-amino-1-[(2R,5S)-2-(hydroxymethyl)-1,3-oxathiolan-5-yl]pyrimidin-2(1H)-one
MFCD00869739
(-)-1-((2R,5S)-2-(Hydroxymethyl)-1,3-oxathiolan-5-yl)cystosine
4-Amino-1-[(2R,5S)-2-(hydroxymethyl)-1,3-oxathiolan-5-yl]-2(1H)-pyrimidinone
Epivir
4-Amino-1-((2R,5S)-2-(hydroxymethyl)-1,3-oxathiolan-5-yl)pyrimidin-2(1H)-one
3&L-SddC
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