CAS 13422-51-0|Hydroxocobalamin

Introduction:Basic information about CAS 13422-51-0|Hydroxocobalamin, including its chemical name, molecular formula, synonyms, physicochemical properties, and safety information, etc.
Common NameHydroxocobalamin
CAS Number13422-51-0Molecular Weight1346.36
Density/Boiling Point/
Molecular FormulaC62H89CoN13O15PMelting Point200ºC (decomposes)
MSDS/Flash Point/

Names

Namehydroxocobalamin
SynonymMore Synonyms

Hydroxocobalamin BiologicalActivity

DescriptionHydroxocobalamin (Vitamin B12a) is an injectable naturally occurring form of vitamin B12 with a favorable adverse effect profile, used as a dietary supplement in the treatment of vitamin B12 deficiency including pernicious anemia[1][2].
Related CatalogResearch Areas >>Metabolic Disease
Target

Human Endogenous Metabolite

References

[1]. Cheungpasitporn W, et al. High-dose hydroxocobalamin for vasoplegic syndrome causing false blood leak alarm. Clin Kidney J. 2017 Jun;10(3):357-362.  

[2]. Wang H, et al. Oral vitamin B12 versus intramuscular vitamin B12 for vitamin B12 deficiency. Cochrane Database Syst Rev. 2018 Mar 15;3:CD004655.  

[3]. Greenberg SS, et al. Hydroxocobalamin (vitamin B12a) prevents and reverses endotoxin-induced hypotension and mortality in rodents: role of nitric oxide. J Pharmacol Exp Ther. 1995 Apr;273(1):257-65.  

Chemical & Physical Properties

Melting Point200ºC (decomposes)
Molecular FormulaC62H89CoN13O15P
Molecular Weight1346.36
Exact Mass1345.567017
PSA484.10000
LogP6.43870
InChIKeyDQOCFCZRZOAIBN-YHKGLSPZSA-L
SMILESCC1=C2N=C(C=C3N=C(C(C)=C4[N-]C(C)(C5N=C1C(C)(CCC(=O)NCC(C)OP(=O)([O-])OC1C(CO)OC(n6cnc7cc(C)c(C)cc76)C1O)C5CC(N)=O)C(C)(CC(N)=O)C4CCC(N)=O)C(C)(CC(N)=O)C3CCC(N)=O)C(C)(C)C2CCC(N)=O.O.[Co+2]
Storage condition2-8°C
Water Solubilitymethanol: 10 mg/mL at 20 °C, clear, dark red

Toxicological Information

CHEMICAL IDENTIFICATION

RTECS NUMBER :
GG3820000
CHEMICAL NAME :
Cobinamide, dihydroxide, dihydrogen phosphate (ester), mono (inner salt), 3'- ester with 5,6- dimethyl-1-alpha-D-ribofuranosylbenzimidazole
CAS REGISTRY NUMBER :
13422-51-0
LAST UPDATED :
199701
DATA ITEMS CITED :
3
MOLECULAR FORMULA :
C62-H89-Co-N13-O15-P

HEALTH HAZARD DATA

ACUTE TOXICITY DATA

TYPE OF TEST :
LD50 - Lethal dose, 50 percent kill
ROUTE OF EXPOSURE :
Intravenous
SPECIES OBSERVED :
Rodent - mouse
DOSE/DURATION :
>50 mg/kg
TOXIC EFFECTS :
Details of toxic effects not reported other than lethal dose value
REFERENCE :
NIIRDN Drugs in Japan (Ethical Drugs). (Yakugyo Jiho Co., Ltd., Tokyo, Japan) Volume(issue)/page/year: -,867,1990 *** NIOSH STANDARDS DEVELOPMENT AND SURVEILLANCE DATA *** NIOSH OCCUPATIONAL EXPOSURE SURVEY DATA : NOES - National Occupational Exposure Survey (1983) NOES Hazard Code - X3794 No. of Facilities: 7 (estimated) No. of Industries: 1 No. of Occupations: 8 No. of Employees: 3157 (estimated) No. of Female Employees: 1154 (estimated)

Safety Information

Hazard CodesXi
Risk PhrasesR36/37/38
Safety PhrasesS26-S36
RIDADRNONH for all modes of transport
WGK Germany3
RTECSGG3820000

Articles41

More Articles
Pseudo-blood leak? A hemodialysis mystery.

Clin. Nephrol. 79(4) , 323-5, (2013)

Hydroxocobalamin is a treatment for cyanide toxicity with few side effects. We report a case of a hemodialysis patient whose treatment was compromised by hydroxocobalamin interference with the blood l...

A patient with an inborn error of vitamin B12 metabolism (cblF) detected by newborn screening.

Pediatrics 132(1) , e257-61, (2013)

A neonate, who was found to have an elevated C3/C2 ratio and minimally elevated propionylcarnitine on newborn screening, was subsequently identified as having the rare cblF inborn error of vitamin B12...

Severe combined immunodeficiency resulting from mutations in MTHFD1.

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Folate and vitamin B(12) metabolism are essential for de novo purine synthesis, and several defects in these pathways have been associated with immunodeficiency. Here we describe the occurrence of sev...

Synonyms

Hydroxocobalamin
Vitamin B12a acetate
EINECS 236-533-2
hydroxycobalamin
ohb12
vitamin B12a
duradoce
cobalex
docevita
MFCD00082532
docclan
hydroxycobalamine
docelan
vibeden
hydrovit
axlon
axion
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